Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 13 hits in this display
BDBM82487(TMQ, 3',5'-Diiodo)
BDBM82487(TMQ, 3',5'-Diiodo)
BDBM82487(TMQ, 3',5'-Diiodo)
BDBM82487(TMQ, 3',5'-Diiodo)
BDBM82487(TMQ, 3',5'-Diiodo)
Ki: 2nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
BDBM82487(TMQ, 3',5'-Diiodo)
BDBM82487(TMQ, 3',5'-Diiodo)
BDBM82487(TMQ, 3',5'-Diiodo)
BDBM82487(TMQ, 3',5'-Diiodo)
Ki: 21nMAssay Description:Binding Affinity against human Beta-3 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
BDBM82487(TMQ, 3',5'-Diiodo)
Ki: 47nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
BDBM82487(TMQ, 3',5'-Diiodo)
BDBM82487(TMQ, 3',5'-Diiodo)
Ki: 79nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
BDBM82487(TMQ, 3',5'-Diiodo)
Ki: 79.4nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair