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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  0.580nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  0.970nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  2nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  2.81nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  5.24nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  21nMAssay Description:Binding Affinity against human Beta-3 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  47nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  79nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  79nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)
Affinity DataKi:  79.4nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed