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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]MDL from rat 5HT2A receptor expressed in GF62 cells by liquid scintillation analyserMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi:  1.84E+3nMAssay Description:Inhibition of human cloned 5HT2B receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi:  3.42E+3nMAssay Description:Inhibition of human cloned 5HT1D receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi:  5.17E+3nMAssay Description:Inhibition of human cloned 5HT7 receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT1B receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT1E receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT3 receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT1A receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT6 receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5HT5A receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Institute Of Nuclear Chemistry Johannes Gutenberg-University Mainz

Curated by ChEMBL
LigandPNGBDBM50267509((3-(2-Fluorethoxy)-2-methoxyphenyl)-(1-(2-p-nitrop...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human cloned 5-HT2C receptor by competitive binding experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed