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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetAurora kinase B(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PIM2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Uit - The Arctic University Of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed