Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  10.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  33.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  44.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  45nMAssay Description:Binding affinity against Beta-2 adrenergic receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  67.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  75.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataKi:  76nMAssay Description:Binding affinity against Beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibitory activity against U-46,619-induced responses in human platelet aggregation (Thromboxane A2 alpha receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataEC50:  240nMAssay Description:Inhibitory activity against Beta-1 adrenergic receptor in guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82482(TMQ, S-(+)-8-Fluoro)
Affinity DataEC50:  295nMAssay Description:Inhibitory activity against Beta-2 adrenergic receptor in guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed