Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  372nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  372nMAssay Description:Binding affinity against Beta-2 adrenergic receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  417nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  417nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  437nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity against Beta-1 adrenergic receptor in guinea pig left ventricleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataKi:  1.15E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataIC50:  2.46E+3nMAssay Description:Inhibitory activity against U-46,619-induced responses in human platelet aggregation (Thromboxane A2 alpha receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataEC50:  3.55E+3nMAssay Description:Inhibitory activity against Beta-2 adrenergic receptor in guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by ChEMBL
LigandPNGBDBM82497(TMQ, R-(-)-8-Fluoro)
Affinity DataEC50:  6.03E+3nMAssay Description:Inhibitory activity against Beta-1 adrenergic receptor in guinea pig atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed