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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
G protein-coupled receptor kinase 5
(Homo sapiens (Human))
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50529465
(CHEMBL4464632)
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Affinity Data
IC50: 220nM
Assay Description:
Inhibition of human GRK5 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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PC cid
PC sid
In Depth
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Article
PubMed
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Target
G protein-coupled receptor kinase 5
(Homo sapiens (Human))
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50529465
(CHEMBL4464632)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6.20E+3nM
Assay Description:
Inhibition of human GRK5 using tubulin as substrate measured after 60 mins by [gamma-32P]-ATP assay
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G protein-coupled receptor kinase 5
(Homo sapiens (Human))
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50529465
(CHEMBL4464632)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.13E+4nM
Assay Description:
Inhibition of human GRK5 using tubulin as substrate measured after 30 mins by [gamma-32P]-ATP assay
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G protein-coupled receptor kinase 5
(Homo sapiens (Human))
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50529465
(CHEMBL4464632)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.90E+4nM
Assay Description:
Inhibition of human GRK5 using tubulin as substrate measured after 0 mins by [gamma-32P]-ATP assay
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Beta-adrenergic receptor kinase 1
(Bos taurus)
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50529465
(CHEMBL4464632)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of bovine GRK2 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay
More data for this Ligand-Target Pair
Target Info
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Ligand Info
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In Depth
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Article
PubMed
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Target
Rhodopsin kinase GRK1
(Bos taurus)
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50529465
(CHEMBL4464632)
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Copy InChI
Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of bovine GRK1 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G protein-coupled receptor kinase 5
(Bos taurus)
University Of Michigan
Curated by
ChEMBL
Ligand
BDBM50529465
(CHEMBL4464632)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.00E+5nM
Assay Description:
Inhibition of bovine GRK5 C474S mutant using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI