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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50336458((3S,5R)-5-bromo-16-hydroxy-14-methoxy-3-methyl-3,4...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human recombinant PDGFRalpha in cell free system after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50336458((3S,5R)-5-bromo-16-hydroxy-14-methoxy-3-methyl-3,4...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human recombinant FLT-3 kinase expressed in insect cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50336458((3S,5R)-5-bromo-16-hydroxy-14-methoxy-3-methyl-3,4...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human recombinant VEGFR2 expressed in Sf9 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50336458((3S,5R)-5-bromo-16-hydroxy-14-methoxy-3-methyl-3,4...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of human recombinant VEGFR3 in cell free system after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50336458((3S,5R)-5-bromo-16-hydroxy-14-methoxy-3-methyl-3,4...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human recombinant c-kit kinase in cell free system after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
National University Of Ireland

Curated by ChEMBL
LigandPNGBDBM50336458((3S,5R)-5-bromo-16-hydroxy-14-methoxy-3-methyl-3,4...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant VEGFR1 expressed in Sf9 cells after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed