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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
11
hits in this display
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
IC50: 520nM
Assay Description:
Inhibition of BRD4 in poly(I:C)-stimulated human SAECs TLR3-inducible CIG5 gene expression pre-incubated for 24 hrs before poly(I:C) stimulation for ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.10E+3nM
Assay Description:
Inhibition of BRD4 in poly(I:C)-stimulated human SAECs TLR3-inducible IL-6 gene expression pre-incubated for 24 hrs before poly(I:C) stimulation for ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
Kd: 684nM
Assay Description:
Binding affinity to recombinant BRD4 BD2 (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 3
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
Kd: 2.40E+3nM
Assay Description:
Binding affinity to recombinant BRD3 BD1 (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
CREB-binding protein
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
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Copy InChI
Affinity Data
Kd: >1.00E+4nM
Assay Description:
Binding affinity to recombinant CBP (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 3
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
Kd: 2.08E+3nM
Assay Description:
Binding affinity to recombinant BRD3 BD2 (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
Kd: 67nM
Assay Description:
Binding affinity to recombinant BRD4 BD1 (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 2
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
Kd: 791nM
Assay Description:
Binding affinity to recombinant BRD2 BD1 (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain testis-specific protein
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
Kd: 2.87E+3nM
Assay Description:
Binding affinity to recombinant BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain-containing protein 2
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
Kd: 845nM
Assay Description:
Binding affinity to recombinant BRD2 BD2 (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bromodomain testis-specific protein
(Homo sapiens (Human))
University Of Texas Medical Branch
Curated by
ChEMBL
Ligand
BDBM50527821
(CHEMBL4455209)
Copy SMILES
Copy InChI
Affinity Data
Kd: 2.32E+3nM
Assay Description:
Binding affinity to recombinant BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI