Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM50085526((E)-3,5,30,40-Tetramethoxystilbene | 4-[(E)-2-(3,5...)
BDBM50085526((E)-3,5,30,40-Tetramethoxystilbene | 4-[(E)-2-(3,5...)
IC50: 160nMAssay Description:Inhibition of wildtype ABCG2 (unknown origin) transfected in HEK293 cells measured after 30 mins by flow cytometric anlaysisMore data for this Ligand-Target Pair
BDBM50085526((E)-3,5,30,40-Tetramethoxystilbene | 4-[(E)-2-(3,5...)
IC50: 750nMAssay Description:Inhibition of ethoxyresorufin O-deethylation (EROD) in bicistronic bacterial membranes epressing human cytochrome P450 1A1More data for this Ligand-Target Pair
BDBM50085526((E)-3,5,30,40-Tetramethoxystilbene | 4-[(E)-2-(3,5...)
IC50: 3.00E+3nMAssay Description:Inhibition of ethoxyresorufin O-deethylation (EROD) in bicistronic bacterial membranes expressing human cytochrome P450 1B1More data for this Ligand-Target Pair
BDBM50085526((E)-3,5,30,40-Tetramethoxystilbene | 4-[(E)-2-(3,5...)
IC50: 3.71E+4nMAssay Description:Inhibition of human quinone reductase 2 expressed in Escherichia coli BL21(DE3) using N-methyldihydronicotinamide as co-substrateMore data for this Ligand-Target Pair
BDBM50085526((E)-3,5,30,40-Tetramethoxystilbene | 4-[(E)-2-(3,5...)
IC50: 5.70E+5nMAssay Description:Inhibition of ethoxyresorufin O-deethylation (EROD) in bicistronic bacterial membranes expressing human cytochrome P450 1A2More data for this Ligand-Target Pair