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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Fibroblast growth factor receptor 2 [403-822]
(Homo sapiens (Human))
Array Biopharma
US Patent
Ligand
BDBM350049
(6-(3-amino-6-(1-methyl- 1H-pyrazol-4-yl)pyrazin- 2...)
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Affinity Data
IC50: 1nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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Target
Fibroblast growth factor receptor 2
(Homo sapiens (Human))
Array Biopharma
US Patent
Ligand
BDBM350049
(6-(3-amino-6-(1-methyl- 1H-pyrazol-4-yl)pyrazin- 2...)
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Copy InChI
Affinity Data
IC50: 1nM
Assay Description:
FGFR1, 2 and 3 kinase activity was measured by the Invitrogen LanthaScreen™ Assay technology which directly measures the amount of substrate phosphor...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Fibroblast growth factor receptor 3 [397-806]
(Homo sapiens (Human))
Array Biopharma
US Patent
Ligand
BDBM350049
(6-(3-amino-6-(1-methyl- 1H-pyrazol-4-yl)pyrazin- 2...)
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Affinity Data
IC50: 1.40nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Fibroblast growth factor receptor 3
(Homo sapiens (Human))
Array Biopharma
US Patent
Ligand
BDBM350049
(6-(3-amino-6-(1-methyl- 1H-pyrazol-4-yl)pyrazin- 2...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.40nM
Assay Description:
FGFR1, 2 and 3 kinase activity was measured by the Invitrogen LanthaScreen™ Assay technology which directly measures the amount of substrate phosphor...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Array Biopharma
US Patent
Ligand
BDBM350049
(6-(3-amino-6-(1-methyl- 1H-pyrazol-4-yl)pyrazin- 2...)
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Affinity Data
IC50: 3.10nM
Assay Description:
FGFR1, 2 and 3 kinase activity was measured by the Invitrogen LanthaScreen™ Assay technology which directly measures the amount of substrate phosphor...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Fibroblast growth factor receptor 1 [308-731]
(Homo sapiens (Human))
Array Biopharma
US Patent
Ligand
BDBM350049
(6-(3-amino-6-(1-methyl- 1H-pyrazol-4-yl)pyrazin- 2...)
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Copy InChI
Affinity Data
IC50: 3.10nM
Assay Description:
To measure FGFR1 kinase activity, 200 pM His-tagged recombinant human FGFR1 catalytic domain (amino acids 308-731) (Life Technologies Cat. No. PR4660...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI