Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50538987(CHEMBL4645688)
Affinity DataKi:  30nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50538987(CHEMBL4645688)
Affinity DataKi:  60nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50538987(CHEMBL4645688)
Affinity DataKi:  5.69E+3nMAssay Description:Inhibition of recombinant human HDAC8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50538987(CHEMBL4645688)
Affinity DataKi:  4.92E+4nMAssay Description:Inhibition of recombinant human HDAC4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50538987(CHEMBL4645688)
Affinity DataIC50:  450nMAssay Description:Inhibition of HDAC in human Cal27 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf

Curated by ChEMBL
LigandPNGBDBM50538987(CHEMBL4645688)
Affinity DataIC50:  830nMAssay Description:Inhibition of HDAC in human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed