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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM300905((2S,3R)-3-cyclopropyl-3-((RS)-2-(4-(5-fluoro-2-met...)
Affinity DataEC50:  5.20nMAssay Description:The assay is performed in 384-well format. HEK cells stably expressing human GPR40 are plated at 15,000 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM300905((2S,3R)-3-cyclopropyl-3-((RS)-2-(4-(5-fluoro-2-met...)
Affinity DataEC50:  3.10nMAssay Description:The assay is performed in 384-well format. HEK cells stably expressing human GPR40 are plated at 15,000 cells per well in growth medium (DMEM/10% fet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent