Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM304771(3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-...)
BDBM304770(3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-...)
BDBM304770(3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-...)
IC50: 550nMAssay Description:100 nL of 100× compound dose response curves (serial 3-fold dilutions) in DMSO are stamped using an Echo liquid handling system (Labcyte) into 384-we...More data for this Ligand-Target Pair
BDBM304771(3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-...)
BDBM304770(3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-...)
EC50: 5.50E+4nMAssay Description:NAD(P)H:quinone oxidoreductase 1 (NQO1), also called DT diaphorase, is a homodimeric FAD-containing enzyme that catalyzes obligatory NAD(P)H-dependen...More data for this Ligand-Target Pair
BDBM304770(3-(7-methoxy-1-methyl-1H-benzo[d][1,2,3]triazol-5-...)
EC50: 2.90E+3nMAssay Description:Activation of Nrf2 in human BEAS2B cells assessed as increase in NQO1 enzymatic activity measured after 48 hrs by MTT assayMore data for this Ligand-Target Pair