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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50201579(CHEMBL3963733)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 to 5 mins by Fluo-4AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50201579(CHEMBL3963733)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed