Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 39 hits in this display
BDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM86242(CAS_64645 | NSC_64645 | Tubocurarine,d)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM86242(CAS_64645 | NSC_64645 | Tubocurarine,d)
BDBM86242(CAS_64645 | NSC_64645 | Tubocurarine,d)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
Ki: 9.72E+3nMAssay Description:Binding affinity for nicotinic acetylcholine receptor alpha4-beta2 was evaluated by its ability to inhibit [3H]NIC binding to rat brain membranesMore data for this Ligand-Target Pair
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
BDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
BDBM81458(CAS_57-94-3 | NSC_6000 | d-Tubocurarine)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
IC50: 7.50E+3nMAssay Description:The SKCa-blocking action was assessed by its ability to inhibit the after hyperpolarization (AHP) in cultured rat sympathetic neuronesMore data for this Ligand-Target Pair
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
BDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)