Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human HDAC6 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  61nMAssay Description:Inhibition of human HDAC7 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  72nMAssay Description:Inhibition of human HDAC1 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  94nMAssay Description:Inhibition of human HDAC3 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  103nMAssay Description:Inhibition of human HDAC11 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  109nMAssay Description:Inhibition of human HDAC5 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  118nMAssay Description:Inhibition of human HDAC4 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  123nMAssay Description:Inhibition of human HDAC9 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  136nMAssay Description:Inhibition of human HDAC8 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  190nMAssay Description:Inhibition of human HDAC10 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333093((S)-6-(19-Methoxy-11-oxo-3,13-dioxa-10-azatricyclo...)
Affinity DataIC50:  268nMAssay Description:Inhibition of human HDAC2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed