Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 19 hits in this display
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
Ki: 870nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
Ki: 3.00E+5nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK293 cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
Ki: 3.00E+5nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR expressed in HEK293 cell membranes after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)
BDBM50014648(6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahydro-isoquino...)