Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

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TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Plexxikon

US Patent

LigandBDBM369012(4-(6,7-dimethoxyquinazolin-4-yl)-2- fluoro-aniline...)Copy SMILESCopy InChI

Affinity DataKi:  5.50E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
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