Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetSigma non-opioid intracellular receptor 1(RAT)
Savannah State University

Curated by ChEMBL
LigandPNGBDBM50401674(CHEMBL2205362)
Affinity DataKi:  27.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in rat brain membrane after 2.5 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Savannah State University

Curated by ChEMBL
LigandPNGBDBM50401674(CHEMBL2205362)
Affinity DataKi:  945nMAssay Description:Displacement of [3H]clonidine from alpha2A adrenergic receptor after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Savannah State University

Curated by ChEMBL
LigandPNGBDBM50401674(CHEMBL2205362)
Affinity DataKi:  1.54E+3nMAssay Description:Displacement of [3H]clonidine from alpha2C adrenergic receptor after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Savannah State University

Curated by ChEMBL
LigandPNGBDBM50401674(CHEMBL2205362)
Affinity DataKi:  2.56E+3nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5-HT2A receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Savannah State University

Curated by ChEMBL
LigandPNGBDBM50401674(CHEMBL2205362)
Affinity DataKi:  2.87E+3nMAssay Description:Displacement of [3H]QNB from human recombinant M4 receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Savannah State University

Curated by ChEMBL
LigandPNGBDBM50401674(CHEMBL2205362)
Affinity DataKi:  7.61E+3nMAssay Description:Displacement of [3H]LY278584 from human recombinant 5-HT3 receptor after 1.5 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed