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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
68
hits in this display
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
Ki: 2.60nM
Assay Description:
Displacement of [3H]CGP12177 from human beta2 adrenoceptor
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
Copy InChI
Affinity Data
Ki: 2.60nM
Assay Description:
Displacement of [125I]iodo-(+/-)-cyanopindolol from human adrenergic beta2 receptor expressed in CHO cells after 3 hrs by radio-ligand binding assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
Ki: 2.60nM
Assay Description:
Binding affinity for human beta-2 adrenergic receptor
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Copy InChI
Affinity Data
Ki: 23nM
Assay Description:
Displacement of [125I]cyanopindolol from human recombinant beta2 adrenergic receptor expressed in CHO cells by filtration assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 26nM
Assay Description:
Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cells
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
Ki: 32nM
Assay Description:
Displacement of [3H]dihydroalprenolol from beta2 receptor (unknown origin) by liquid scintillation counting and cell based assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
Ki: 32nM
Assay Description:
Displacement of [3H]dihydroalprenolol from human beta2 adrenergic receptor expressing cell membrane by competition binding assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
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Affinity Data
Ki: 33nM
Assay Description:
Displacement of [3H]-dihydroalprenolol from human beta2-adrenoceptor expressed in HEK cells after 4 hrs
Checked by Author
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
Ki: 315nM
Assay Description:
Displacement of [125I]iodo-(+/-)-cyanopindolol from human adrenergic beta1 receptor expressed in CHO cells after 3 hrs by radio-ligand binding assay
More data for this Ligand-Target Pair
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
Copy InChI
Affinity Data
Ki: 319nM
Assay Description:
Displacement of [3H]CGP12177 from human beta-1 adrenoceptor
More data for this Ligand-Target Pair
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
Ki: 1.63E+3nM
Assay Description:
Displacement of [125I]7-HO-PIPAT from human D3R expressed in HEK cells
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
Ki: 1.71E+3nM
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
Ki: 2.00E+3nM
Assay Description:
Displacement of [3H]dihydroalprenolol from beta1 receptor (unknown origin) by liquid scintillation counting and cell based assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
Ki: 2.57E+3nM
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Target
Beta-3 adrenergic receptor
(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by
PDSP K
i
Database
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
Ki: 8.09E+3nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Affinity Data
Ki: 1.30E+4nM
Assay Description:
Displacement of [3H]spiperone from human D2S receptor expressed in CHO cells
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Affinity Data
IC50: 0.400nM
Assay Description:
Agonist activity at beta2 adrenergic receptor in guinea pig tracheal strip assessed as inhibition of electrically-induced bronchocontractile response...
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
IC50: 0.400nM
Assay Description:
Agonist activity at adrenergic beta2 receptor in electrically-stimulated Dunkin-Hartley guinea pig tracheal strip assessed as inhibition of contracti...
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
IC50: <631nM
Assay Description:
Binding affinity to adrenergic beta1 receptor
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
IC50: <631nM
Assay Description:
Binding affinity to beta1 adrenoceptor
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
Friedrich-Alexander University
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
IC50: <1.00E+4nM
Assay Description:
Binding affinity to dopamine 2 receptor
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Target
ATP-binding cassette sub-family C member 3
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP3 overexpressed in Sf9 insect cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ...
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Target
ATP-binding cassette sub-family C member 4
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...
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Target
Bile salt export pump
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...
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Target
ATP-binding cassette sub-family C member 2
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
IC50: >1.33E+5nM
Assay Description:
Inhibition of human MRP2 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...
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Target
Orotidine 5'-phosphate decarboxylase
(Aspergillus niger)
The Scripps Research Institute Molecular Screening Center
Curated by
PubChem BioAssay
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Affinity Data
EC50: >5.96E+4nM
Assay Description:
Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRISMC) Center Affiliation: The Scripps Research Institute, TS...
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Affinity Data
EC50: 1.30nM
Assay Description:
Agonist activity at human beta2 adrenergic receptor assessed as increase in cAMP level by whole cell assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
EC50: 0.501nM
Assay Description:
Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...
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Target
Beta-3 adrenergic receptor
(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by
PDSP K
i
Database
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
EC50: 40nM
Assay Description:
Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-g...
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Target
Beta-1 adrenergic receptor
(GUINEA PIG)
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
EC50: 0.316nM
Assay Description:
Agonist activity at beta-1 adrenergic receptor in guinea pig trachea assessed as inhibition of electrical stimulation-induced muscle contraction
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
EC50: 1.60nM
Assay Description:
Agonist activity at beta2 receptor in guinea pig trachea assessed as fast onset of inhibition of electrically stimulated contraction
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
EC50: 13nM
Assay Description:
Agonist activity at human recombinant beta1 receptor assessed as cAMP accumulation by radioimmunoassay and cell based assay
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Target
Beta-3 adrenergic receptor
(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by
PDSP K
i
Database
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human recombinant beta3 receptor assessed as cAMP accumulation by radioimmunoassay and cell based assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
EC50: 2.5nM
Assay Description:
Agonist activity at human beta2 receptor in BEAS-2B cells assessed as cAMP accumulation by radioimmunoassay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
EC50: 0.200nM
Assay Description:
Agonist activity at human recombinant beta2 receptor assessed as cAMP accumulation by radioimmunoassay and cell based assay
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Copy BDB DOI
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
EC50: 2.5nM
Assay Description:
Agonist activity at human beta2 adrenergic receptor in human BEAS-2B cells by cAMP accumulation assay
More data for this Ligand-Target Pair
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Copy BDB DOI
Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
EC50: 13nM
Assay Description:
Agonist activity at human beta1 adrenergic receptor expressed in cells by cAMP accumulation assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.200nM
Assay Description:
Agonist activity at human beta2 adrenergic receptor expressed in cells by cAMP accumulation assay
More data for this Ligand-Target Pair
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Target
Beta-3 adrenergic receptor
(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by
PDSP K
i
Database
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human beta3 adrenergic receptor expressed in cells by cAMP accumulation assay
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Affinity Data
EC50: 0.400nM
Assay Description:
Agonist activity at human adrenergic beta 2 expressed in CHO-K1 cells assessed as intracellular cAMP accumulation
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Copy BDB DOI
Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
Copy InChI
Affinity Data
EC50: 86nM
Assay Description:
Agonist activity at human recombinant adrenergic beta-1 receptor expressed in CHO cells assessed as cAMP accumulation
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.400nM
Assay Description:
Agonist activity at human recombinant adrenergic beta2 receptor expressed in CHO cells assessed as cAMP accumulation
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.400nM
Assay Description:
Agonist activity at human beta2 adrenoceptor expressed in CHOK1 cell assessed as increase of intracellular cAMP level
More data for this Ligand-Target Pair
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Copy BDB DOI
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
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Affinity Data
EC50: 7.90nM
Assay Description:
Agonist activity at beta 2 in human A431 cells adrenoceptor assessed as cAMP accumulation
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.501nM
Assay Description:
Agonist activity at human recombinant beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation after...
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Copy BDB DOI
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.501nM
Assay Description:
Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as intracellular cAMP accumulation after 1 hr
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1nM
Assay Description:
Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as stimulation of cAMP accumulation after 60 mins
More data for this Ligand-Target Pair
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.501nM
Assay Description:
Agonist activity at human adrenergic beta2 receptor expressed in CHO cells assessed as cAMP accumulation
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.501nM
Assay Description:
Agonist activity at human beta2 receptor expressed in CHO cells assessed as cAMP accumulation
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1nM
Assay Description:
Agonist activity at human beta2 adrenoceptor expressed in H292 cells assessed as increase in cAMP accumulation after 60 mins by spectrophotometry
More data for this Ligand-Target Pair
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 86nM
Assay Description:
Agonist activity at human beta-1 adrenoceptor expressed in CHOK1 cell assessed as increase of intracellular cAMP level
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 86nM
Assay Description:
Agonist activity at human adrenergic beta 1 expressed in CHO-K1 cells assessed as intracellular cAMP accumulation
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
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Affinity Data
EC50: 0.190nM
Assay Description:
Agonist activity at human beta2-adrenoceptor expressed in HEK cells assessed as increase of cAMP level after 10 mins by radioimmuno assay
Checked by Author
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Affinity Data
EC50: 0.126nM
Assay Description:
Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contraction
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.130nM
Assay Description:
Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contraction
More data for this Ligand-Target Pair
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.126nM
Assay Description:
Agonist activity at beta2 adrenoceptor in guinea pig assessed as relaxation of histamine-induced tracheal ring contraction
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 40nM
Assay Description:
Agonist activity at human adrenergic beta1 receptor expressed in CHO cells assessed as cAMP accumulation
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Target
Beta-3 adrenergic receptor
(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by
PDSP K
i
Database
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human adrenergic beta3 receptor expressed in CHO cells assessed as cAMP accumulation
More data for this Ligand-Target Pair
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.316nM
Assay Description:
Agonist activity at adrenergic beta2 receptor in guinea pig trachea assessed as inhibition of electrically-stimulated contraction
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 40nM
Assay Description:
Agonist activity at human beta1 receptor expressed in CHO cells assessed as cAMP accumulation
More data for this Ligand-Target Pair
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Target
Beta-2 adrenergic receptor
(GUINEA PIG)
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.316nM
Assay Description:
Agonist activity at beta2 adrenergic receptor in guinea pig tracheal strip assessed as inhibition of electrically-induced bronchocontractile response
More data for this Ligand-Target Pair
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Target
Beta-3 adrenergic receptor
(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by
PDSP K
i
Database
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human beta3 receptor expressed in CHO cells assessed as cAMP accumulation
More data for this Ligand-Target Pair
Target Info
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antibodypedia
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Target
Beta-3 adrenergic receptor
(Homo sapiens (Human))
UniversitÄT WÜRzburg
Curated by
PDSP K
i
Database
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 25nM
Assay Description:
Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation after...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
Ligand Info
Purchase
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Article
PubMed
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Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
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Affinity Data
EC50: 40nM
Assay Description:
Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation afte...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
Ligand Info
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Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM86453
(CAS_73573-87-2 | Formoterol | NSC_3083544)
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Affinity Data
Kd: 2.5nM
Assay Description:
Binding affinity to beta-2 adrenergic receptor (unknown origin) at 1 to 10000 nM
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
UniProtKB/SwissProt
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antibodypedia
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Copy BDB DOI
Target
Beta-1 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 109nM
Assay Description:
Agonist activity at human beta1 adrenoceptor expressed in CHO cells assessed as increase in intracellular cAMP level incubated for 1 hr by alphascree...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
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Article
PubMed
Copy BDB DOI
Target
Beta-2 adrenergic receptor
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50151720
(ARFORMOTEROL TARTRATE | CHEMBL1363 | CHEMBL605993 ...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2.60nM
Assay Description:
Agonist activity at human beta2 adrenoceptor expressed in CHO cells assessed as increase in intracellular cAMP level incubated for 1 hr by alphascree...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
CHEMBL
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MCE
KEGG
PC cid
PC sid
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Article
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3D Structure (crystal)
Copy BDB DOI
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