Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Janssen Research & Developmen

Curated by ChEMBL

LigandBDBM50548189(CHEMBL4761101)Copy SMILESCopy InChI

Affinity DataEC50:  9.40nMAssay Description:Agonist activity at human GPR40 transfected in HEK293 cells assessed as increase in intracellular calcium level incubated for 1 hr by Fluo-8 dye base...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMelanocortin receptor 4(Rattus norvegicus)
Janssen Research & Developmen

Curated by ChEMBL

LigandBDBM50548189(CHEMBL4761101)Copy SMILESCopy InChI

Affinity DataEC50:  45nMAssay Description:Agonist activity at rat GPR40 transfected in HEK293 cells assessed as increase in intracellular calcium level incubated for 1 hr by Fluo-8 dye based ...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI