Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetFree fatty acid receptor 1(Homo sapiens (Human))TBA

LigandBDBM50244024(CHEMBL4081072)Copy SMILESCopy InChI

Affinity DataEC50:  210nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails PubMed
Copy BDB DOI

TargetFree fatty acid receptor 1(Homo sapiens (Human))TBA

LigandBDBM50244024(CHEMBL4081072)Copy SMILESCopy InChI

Affinity DataEC50:  210nMAssay Description:Agonist activity at human GPR40 expressed in CHOA12 cells assessed as induction of Ca2+ mobilization by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI