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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Protein O-GlcNAcase
(Homo sapiens (Human))
University Of Debrecen
Curated by
ChEMBL
Ligand
BDBM50577839
(CHEMBL4851727)
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Affinity Data
Ki: 270nM
Assay Description:
Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Beta-hexosaminidase
(Bos taurus)
University Of Debrecen
Curated by
ChEMBL
Ligand
BDBM50577839
(CHEMBL4851727)
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Copy InChI
Affinity Data
Ki: 413nM
Assay Description:
Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI