Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113676((S)-benzyl 1-(2-(4-methoxyphenylamino)ethylamino)-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113676((S)-benzyl 1-(2-(4-methoxyphenylamino)ethylamino)-...)
Affinity DataIC50:  70nMAssay Description:Inhibitory activity against recombinant human cathepsin K activity using fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113676((S)-benzyl 1-(2-(4-methoxyphenylamino)ethylamino)-...)
Affinity DataIC50:  90nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50113676((S)-benzyl 1-(2-(4-methoxyphenylamino)ethylamino)-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin S activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50113676((S)-benzyl 1-(2-(4-methoxyphenylamino)ethylamino)-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory activity against recombinant human cathepsin L activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed