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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataKi:  11nMAssay Description:Eq. constant (Ki) for inhibition of Cathepsin K was determined by progress curves, following hydrolysis of Z-Phe-Arg- Amc in the absence and presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human cathepsin K in fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant human cathepsin S in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed