Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetBeta-2 adrenergic receptor(GUINEA PIG)
Theravance

Curated by ChEMBL
LigandPNGBDBM50018588(CHEMBL3290998)
Affinity DataEC50:  13nMAssay Description:Agonist activity at beta2 receptor in guinea pig trachea assessed as slow onset of inhibition of electrically stimulated contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50018588(CHEMBL3290998)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant beta1 receptor assessed as cAMP accumulation by radioimmunoassay and cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50018588(CHEMBL3290998)
Affinity DataEC50:  0.126nMAssay Description:Agonist activity at human recombinant beta2 receptor assessed as cAMP accumulation by radioimmunoassay and cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50018588(CHEMBL3290998)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at human beta2 receptor in BEAS-2B cells assessed as cAMP accumulation by radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Theravance

Curated by ChEMBL
LigandPNGBDBM50018588(CHEMBL3290998)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at human recombinant beta3 receptor assessed as cAMP accumulation by radioimmunoassay and cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed