Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetHistone deacetylase 2(Homo sapiens (Human))
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM347457(US9790158, 8)
Affinity DataKi:  0.510nMAssay Description:Inhibition of human recombinant HDAC2 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Connecticut

US Patent
LigandPNGBDBM347457(US9790158, 8)
Affinity DataKi:  1.42nMAssay Description:Key enzyme kinetic parameters for one class I HDAC (HDAC8) and one class Ha HDAC (HDAC4) were determined using commercially available human recombina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Connecticut

US Patent
LigandPNGBDBM347457(US9790158, 8)
Affinity DataKi:  266nMAssay Description:Inhibition of human recombinant HDAC8 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
University of Connecticut

US Patent
LigandPNGBDBM347457(US9790158, 8)
Affinity DataKi:  541nMAssay Description:Key enzyme kinetic parameters for one class I HDAC (HDAC8) and one class Ha HDAC (HDAC4) were determined using commercially available human recombina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM347457(US9790158, 8)
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of human recombinant HDAC1 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM347457(US9790158, 8)
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of human recombinant HDAC6 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM347457(US9790158, 8)
Affinity DataKi: >2.50E+3nMAssay Description:Inhibition of human recombinant HDAC5 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
University of Connecticut

US Patent
LigandPNGBDBM347457(US9790158, 8)
Affinity DataKi:  1.12E+4nMAssay Description:Inhibition of human recombinant HDAC4 by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed