Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50:  50nMAssay Description:For the enzyme assay, the enzyme fraction was added to fluorescent substrate in the presence of test compounds, and the mixture was incubated for add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Methylgene

LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant HDAC1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50:  200nMAssay Description:Inhibition of recombinant HDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50:  200nMAssay Description:For the enzyme assay, the enzyme fraction was added to fluorescent substrate in the presence of test compounds, and the mixture was incubated for add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant HDAC3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant HDAC6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Methylgene

LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: >2.00E+4nMAssay Description:For the enzyme assay, the enzyme fraction was added to fluorescent substrate in the presence of test compounds, and the mixture was incubated for add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: >2.00E+4nMAssay Description:For the enzyme assay, the enzyme fraction was added to fluorescent substrate in the presence of test compounds, and the mixture was incubated for add...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Methylgene

LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant HDAC8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed