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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProteasome subunit beta type-8(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM388354(US10294246, Compound No. 51 | [(1R)-2-(benzofuran-...)
Affinity DataIC50: <50nMAssay Description:Measurement of LMP7 inhibition is performed in 384 well format based on fluorescence intensity assay.Purified human immunoproteasome (0.25 nM) and se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Merck Patent

US Patent
LigandPNGBDBM388354(US10294246, Compound No. 51 | [(1R)-2-(benzofuran-...)
Affinity DataIC50:  2.75E+3nMAssay Description:Measurement of Beta5 inhibition is performed in 384 well format based on fluorescence intensity assay.Purified human constitutive proteasome (1.25 nM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent