Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataKi:  164nMAssay Description:Binding affinity to 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataKi:  392nMAssay Description:Binding affinity to Sigma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataKi:  863nMAssay Description:Binding affinity to alpha1 adrenoreceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  1.98E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  5.77E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  5.80E+3nMAssay Description:Antagonist activity at 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  5.85E+3nMAssay Description:Displacement of [3H]-ketanserin from 5HT2A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Sk Biopharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50393649(CHEMBL2158704)
Affinity DataIC50:  8.82E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed