Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
Kancera

US Patent
LigandPNGBDBM443106(2-[2-fluoro-4-(6-methoxypyridin-3- yl)phenyl]-N-hy...)
Affinity DataIC50:  16nMAssay Description:The assay principle is well known and all necessary reagents like enzymes, substrates, developer and reference compounds are commercially available. ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 8(Homo sapiens (Human))
Kancera

US Patent
LigandPNGBDBM443106(2-[2-fluoro-4-(6-methoxypyridin-3- yl)phenyl]-N-hy...)
Affinity DataIC50:  384nMAssay Description:The assay principle is well known and all necessary reagents like enzymes, substrates, developer and reference compounds are commercially available. ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 3(Homo sapiens (Human))
Kancera

US Patent
LigandPNGBDBM443106(2-[2-fluoro-4-(6-methoxypyridin-3- yl)phenyl]-N-hy...)
Affinity DataIC50:  960nMAssay Description:The assay principle is well known and all necessary reagents like enzymes, substrates, developer and reference compounds are commercially available. ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
Kancera

US Patent
LigandPNGBDBM443106(2-[2-fluoro-4-(6-methoxypyridin-3- yl)phenyl]-N-hy...)
Affinity DataIC50: >2.00E+5nMAssay Description:The assay principle is well known and all necessary reagents like enzymes, substrates, developer and reference compounds are commercially available. ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 2(Homo sapiens (Human))
Kancera

US Patent
LigandPNGBDBM443106(2-[2-fluoro-4-(6-methoxypyridin-3- yl)phenyl]-N-hy...)
Affinity DataIC50: >2.00E+5nMAssay Description:The assay principle is well known and all necessary reagents like enzymes, substrates, developer and reference compounds are commercially available. ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent