Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetHistone deacetylase 7(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50: >10nMAssay Description:Inhibition of recombinant HDAC7 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC as substrate pre-incubated for 1 hr followed by substrate additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50: >10nMAssay Description:Inhibition of recombinant HDAC9 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC as substrate pre-incubated for 1 hr followed by substrate additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50: >10nMAssay Description:Inhibition of recombinant HDAC4 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC as substrate pre-incubated for 1 hr followed by substrate additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant HDAC6 (unknown origin) using Boc-Lys(acetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant HDAC6 (unknown origin) using Boc-Lys(acetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  771nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate pre-incubated for 1 hr followed by substrate addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  776nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using Boc-Lys(Ac)-AMC as substrate pre-incubated for 1 hr followed by substrate addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of recombinant HDAC3 (unknown origin) using Boc-Lys(acetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of recombinant HDAC3 (unknown origin) using Boc-Lys(acetyl)-AMC as substrate preincubated for 1 hr followed by substrate addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  2.82E+3nMAssay Description:Inhibition of recombinant HDAC2 (unknown origin) using Boc-Lys(Ac)-AMC as substrate pre-incubated for 1 hr followed by substrate addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  2.85E+3nMAssay Description:Inhibition of recombinant HDAC2 (unknown origin) using Boc-Lys(Ac)-AMC as substrate pre-incubated for 1 hr followed by substrate addition and measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  3.55E+3nMAssay Description:Inhibition of recombinant HDAC8 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC as substrate pre-incubated for 1 hr followed by substrate additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50581678(CHEMBL5072502)
Affinity DataIC50:  3.59E+3nMAssay Description:Inhibition of recombinant HDAC8 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC as substrate pre-incubated for 1 hr followed by substrate additio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed