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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM49264(MLS000065676 | N-(6-methoxy-1,3-benzothiazol-2-yl)...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM49264(MLS000065676 | N-(6-methoxy-1,3-benzothiazol-2-yl)...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of Photinus pyralis luciferase by PK-Light assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM49264(MLS000065676 | N-(6-methoxy-1,3-benzothiazol-2-yl)...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of Photinus pyralis luciferase by Easy lite assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM49264(MLS000065676 | N-(6-methoxy-1,3-benzothiazol-2-yl)...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of Photinus pyralis luciferase by BrightGlo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM49264(MLS000065676 | N-(6-methoxy-1,3-benzothiazol-2-yl)...)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of Photinus pyralis luciferase by Steady-Glo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor p65(Homo sapiens (Human))
Srmlsc

Curated by PubChem BioAssay
LigandPNGBDBM49264(MLS000065676 | N-(6-methoxy-1,3-benzothiazol-2-yl)...)
Affinity DataEC50:  3.99E+3nMAssay Description:Southern Research Molecular Libraries Screening Center (SRMLSC) Southern Research Institute (Birmingham, Alabama) NIH Molecular Libraries Screening C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay