Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
12
hits in this display
Target
Beta-adrenergic receptor kinase 1
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: 19nM
Assay Description:
Inhibition of human GRK2 by transcreener assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aurora kinase A
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: 137nM
Assay Description:
Inhibition of human Aurora A
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Rho-associated protein kinase 1
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.27E+3nM
Assay Description:
Inhibition of human ROCK1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Ribosomal protein S6 kinase alpha-1
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.15E+3nM
Assay Description:
Inhibition of RSK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Rhodopsin kinase GRK7
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human GRK7
More data for this Ligand-Target Pair
Target Info
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Protein kinase C beta type
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human PKCbeta1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Calcium/calmodulin-dependent protein kinase type II subunit beta
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human CaMK2beta
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G protein-coupled receptor kinase 5
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human GRK5
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Rhodopsin kinase GRK1
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human GRK1
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Protein kinase C alpha type
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human PKCalpha
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human PKBalpha
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
G protein-coupled receptor kinase 6
(Homo sapiens (Human))
Janssen Research & Development
Curated by
ChEMBL
Ligand
BDBM50554258
(CHEMBL4744858)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of human GRK6
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI