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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetChromobox protein homolog 7(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515921(CHEMBL4551668)
Affinity DataKd:  5.30E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged CBX7 (1 to 62 residues) expressed in Escherichia coli BL2 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromodomain Y-like protein 2(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515921(CHEMBL4551668)
Affinity DataKd:  3.58E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged CDYL2 (1 to 70 residues) expressed in Escherichia coli BL2 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromodomain Y-like protein(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515921(CHEMBL4551668)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged CDYL (1 to 60 residues) expressed in Escherichia coli BL2 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTestis-specific chromodomain protein Y 1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515921(CHEMBL4551668)
Affinity DataKd:  1.13E+4nMAssay Description:Binding affinity to recombinant human N-terminal GST-tagged CDY1 (1 to 65 residues) expressed in Escherichia coli BL2 by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed