Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

LigandPNGBDBM50267196((+/-)1-(1H-indol-4-yloxy)-3-(2-(2-methoxyphenoxy)e...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]Clonidine from alpha2 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
RzeszóW University Of Technology

Curated by ChEMBL
LigandPNGBDBM50267197((2S)-1-(1H-Indol-4-yloxy)-3-{[2-(2-methoxyphenoxy)...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
RzeszóW University Of Technology

Curated by ChEMBL
LigandPNGBDBM50267196((+/-)1-(1H-indol-4-yloxy)-3-(2-(2-methoxyphenoxy)e...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Rzesz£W University Of Technology

Curated by ChEMBL
LigandPNGBDBM50267196((+/-)1-(1H-indol-4-yloxy)-3-(2-(2-methoxyphenoxy)e...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]Prazosin from alpha1 adrenergic receptor in Wistar rat cerebral cortex membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
RzeszóW University Of Technology

Curated by ChEMBL
LigandPNGBDBM50267198((2R)-1-(1H-Indol-4-yloxy)-3-{[2-(2-methoxyphenoxy)...)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]CGP12177 from beta1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed