Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM314379(US9611261, Example 2b-A | US9611261, Example 2b-B ...)
BDBM314379(US9611261, Example 2b-A | US9611261, Example 2b-B ...)
IC50: 604nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
BDBM314379(US9611261, Example 2b-A | US9611261, Example 2b-B ...)
IC50: 4.12E+4nMAssay Description:The assay buffer used in this screen is 0.05 M acetate, pH 4.2, 10% DMSO final, 100 uM genapol (which is a nonionic detergent, below its Critical Mic...More data for this Ligand-Target Pair
BDBM314379(US9611261, Example 2b-A | US9611261, Example 2b-B ...)
BDBM314379(US9611261, Example 2b-A | US9611261, Example 2b-B ...)
IC50: 8.13E+4nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair
BDBM314379(US9611261, Example 2b-A | US9611261, Example 2b-B ...)
IC50: >4.00E+5nMAssay Description:Recombinant Cat D was expressed in CHO cells. The assay buffer for CathepsinD is 0.05 M citrate pH 3.5, 10% DMSO final, 5 mM CHAPS. The Cat D enzyme ...More data for this Ligand-Target Pair