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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50001909(CHEMBL163153 | N-(4-{[(4-Phenyl-piperazin-2-ylmeth...)
Affinity DataIC50:  3.00E+3nMAssay Description:Binding affinity for Beta-1 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine ventricular...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Canis familiaris)
Berlex Laboratories

Curated by ChEMBL
LigandPNGBDBM50001909(CHEMBL163153 | N-(4-{[(4-Phenyl-piperazin-2-ylmeth...)
Affinity DataIC50:  4.60E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed