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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 40 hits in this display   

TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human recombinant DPP4 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by manual whole-cell patch-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50:  4.58E+4nMAssay Description:Inhibition of recombinant human CYP3A4 using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50:  4.58E+4nMAssay Description:Inhibition of recombinant human CYP3A5 using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50:  7.63E+4nMAssay Description:Inhibition of recombinant human CYP2C8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2B6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2A6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using testosterone as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using testosterone as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2E1(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2E1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2B6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2A6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using testosterone as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using testosterone as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2E1(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2E1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2B6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2A6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DPP9 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DPP8 incubated for 15 mins using Gly-Pro-7-AMC substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2E1(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2E1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A4 using testosterone as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP3A5 using testosterone as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Haisco Pharmaceutical Group

Curated by ChEMBL
LigandPNGBDBM50540846(CHEMBL4646510)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human CYP2C19More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed