Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 22 hits in this display
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
EC50: 1.00E+5nMAssay Description:The compound was evaluated for agonist activity against phospholipase C coupled recombinant human P2Y purinoceptor 6 (P2Y6)More data for this Ligand-Target Pair
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
EC50: 4.5nMAssay Description:Agonists activity was evaluated by release of [Ca2+] release of HEK 293 cells stably transfected with rat-brain P2Y purinoceptor 1 (P2Y1-R)More data for this Ligand-Target Pair
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
EC50: 1.50E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat receptor P2X purinoceptor 2 (P2X2) at 10 uM, expressed in Xenopus oocytesMore data for this Ligand-Target Pair
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
EC50: 5.00E+4nMAssay Description:The compound was evaluated for antagonist activity against phospholipase C coupled human P2Y purinoceptor 11 (P2Y11)More data for this Ligand-Target Pair
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
EC50: 350nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 3 (P2X3) at 10 uM, expressed in Xenopus oocytesMore data for this Ligand-Target Pair
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)
BDBM50118232(2-MeSATP | ATP, 2-meS | CHEMBL336208)