Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Allergan

Curated by ChEMBL

LigandBDBM50055829((1H-Imidazol-2-yl)-(5-methyl-quinoxalin-6-yl)-amin...)Copy SMILESCopy InChI

Affinity DataKi:  31nMAssay Description:Displacement of rauwolscine from human Alpha-2A adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Allergan

Curated by ChEMBL

LigandBDBM50055829((1H-Imidazol-2-yl)-(5-methyl-quinoxalin-6-yl)-amin...)Copy SMILESCopy InChI

Affinity DataKi:  340nMAssay Description:Displacement of rauwolscine from human Alpha-2C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Allergan

Curated by ChEMBL

LigandBDBM50055829((1H-Imidazol-2-yl)-(5-methyl-quinoxalin-6-yl)-amin...)Copy SMILESCopy InChI

Affinity DataKi:  1.20E+3nMAssay Description:Displacement of rauwolscine from rat Alpha-2B adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
Copy BDB DOI