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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCoagulation factor XII(Homo sapiens (Human))
University of Namur

LigandPNGBDBM23566(3-Carboxamide-coumarin deriv., 43 | 6,8-dichloro-N...)
Affinity DataIC50:  4.30E+3nMAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasma kallikrein(Homo sapiens (Human))
University of Namur

LigandPNGBDBM23566(3-Carboxamide-coumarin deriv., 43 | 6,8-dichloro-N...)
Affinity DataIC50: >5.00E+4nMAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
University of Namur

LigandPNGBDBM23566(3-Carboxamide-coumarin deriv., 43 | 6,8-dichloro-N...)
Affinity DataIC50: >5.00E+4nMAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University of Namur

LigandPNGBDBM23566(3-Carboxamide-coumarin deriv., 43 | 6,8-dichloro-N...)
Affinity DataIC50: >5.00E+4nMAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University of Namur

LigandPNGBDBM23566(3-Carboxamide-coumarin deriv., 43 | 6,8-dichloro-N...)
Affinity DataIC50: >5.00E+4nMAssay Description:After substrate hydrolysis reaction, the absorbance at 405 nm was measured in a microplate reader. Percentages of inhibition at each concentration we...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed