Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL

LigandBDBM50566366(CHEMBL4854804)Copy SMILESCopy InChI

Affinity DataEC50:  2.78E+4nMAssay Description:Agonist activity at human PPARgamma expressed in CHO cells assessed as increase in receptor transcriptional activity incubated for 24 hrs by dual luc...More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL

LigandBDBM50566366(CHEMBL4854804)Copy SMILESCopy InChI

Affinity DataEC50:  0.25nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in CHO cells co-expressing luc2P/SRE assessed as firefly luciferase activity incubated for 24 hr...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI