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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Peroxisome proliferator-activated receptor delta
(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation
Curated by
ChEMBL
Ligand
BDBM50312425
(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
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Affinity Data
EC50: 15nM
Assay Description:
Agonist activity at human PPARdelta ligand binding domain by FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor delta
(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation
Curated by
ChEMBL
Ligand
BDBM50312425
(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 10nM
Assay Description:
Agonist activity at human PPARdelta ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor gamma
(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation
Curated by
ChEMBL
Ligand
BDBM50312425
(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Agonist activity at human PPARgamma ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor alpha
(Homo sapiens (Human))
The Genomics Institute Of The Novartis Research Foundation
Curated by
ChEMBL
Ligand
BDBM50312425
(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Agonist activity at human PPARalpha ligand binding domain expressed in human 293T cells cotransfected with Gal4-DBD by luciferase transactivation ass...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor delta
(Mus musculus)
The Genomics Institute Of The Novartis Research Foundation
Curated by
ChEMBL
Ligand
BDBM50312425
(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 31nM
Assay Description:
Agonist activity at mouse PPARdelta by FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI