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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50342692
(4-(1'-(5-chloropyrimidin-2-yl)-4,4'-bipiperidin-1-...)
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Affinity Data
IC50: 277nM
Assay Description:
Inhibition of human ERG
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
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Target
Glucose-dependent insulinotropic receptor
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50342692
(4-(1'-(5-chloropyrimidin-2-yl)-4,4'-bipiperidin-1-...)
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Copy InChI
Affinity Data
EC50: 2nM
Assay Description:
Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glucose-dependent insulinotropic receptor
(Mus musculus)
Merck
Curated by
ChEMBL
Ligand
BDBM50342692
(4-(1'-(5-chloropyrimidin-2-yl)-4,4'-bipiperidin-1-...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 11nM
Assay Description:
Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
In Depth
Details
Article
PubMed
Copy BDB DOI