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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Histone deacetylase 2
(Homo sapiens (Human))
Beijing University Of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50564474
(CHEMBL4795802)
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Affinity Data
IC50: 23nM
Assay Description:
Inhibition of recombinant human HDAC2 using FLUOR-DE-LYS-Green as substrate incubated for 10 mins followed by substrate addition and measured after 3...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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In Depth
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Article
PubMed
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Target
Histone deacetylase 1
(Homo sapiens (Human))
Beijing University Of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50564474
(CHEMBL4795802)
Copy SMILES
Copy InChI
Affinity Data
IC50: 71nM
Assay Description:
Inhibition of recombinant human HDAC1 using SIRT1 as substrate incubated for 10 mins followed by substrate addition and measured after 30 mins by flu...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cyclin-A2/Cyclin-dependent kinase 2
(Homo sapiens (Human))
Beijing University Of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50564474
(CHEMBL4795802)
Copy SMILES
Copy InChI
Affinity Data
IC50: 800nM
Assay Description:
Inhibition of recombinant human N-terminal GST-tagged CDK2/CyclinA2 expressed in baculovirus infected Sf21 cells using histone H1 as substrate incuba...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI