Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Guangdong Pharmaceutical University

Curated by ChEMBL

LigandBDBM50603297(CHEMBL5175597)Copy SMILESCopy InChI

Affinity DataEC50:  3.63E+3nMAssay Description:Agonist activity at pBIND tagged human PPARdelta expressed in human HepG2 cells incubated for 18 hrs by dual luciferase reporter assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
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TargetFree fatty acid receptor 1(Homo sapiens (Human))
Guangdong Pharmaceutical University

Curated by ChEMBL

LigandBDBM50603297(CHEMBL5175597)Copy SMILESCopy InChI

Affinity DataEC50:  1.53E+3nMAssay Description:Agonist activity at human FFA1 expressed in CHO cells assessed as increase in calcium level measured by Fluo-4-AM staining based FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI