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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetFree fatty acid receptor 4(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  471nMAssay Description:Agonist activity at GPR120 (unknown origin) by Fluo-4 AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  43.6nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  95.5nMAssay Description:Agonist activity at GPR120 expressed in Flp-In TREx293 cells by calcium assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Mus musculus)
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  17.0nMAssay Description:Agonist activity at mouse GPR120More data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at FFAR1 expressed in Flp-In TREx293 cells by calcium assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  3.39E+4nMAssay Description:Agonist activity at human FFA1 receptor expressed in CHO-K1 cells assessed as increase in dynamic mass redistribution response by DMR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human FFAR4 expressed in CHO cells assessed as beta-arrestin recruitment after 90 mins by luminescence assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  7.59E+4nMAssay Description:Agonist activity at human FFAR1 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  5.26E+4nMAssay Description:Agonist activity at human FFAR1 expressed in CHO cells assessed as increase in intracellular calcium level by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human FFAR4 expressed in CHO cells assessed as beta-arrestin recruitment after 90 mins by luminescence assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens)
Dalian Institute Of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human FFA4 receptor expressed in CHO-K1 cells assessed as increase in amplitude of dynamic mass redistribution response by DMR as...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  6.46E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed