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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCarbonic anhydrase 9(Homo sapiens (Human))
Egyptian Russian University

Curated by ChEMBL
LigandPNGBDBM50378550(CHEMBL4167551)
Affinity DataKi:  37nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 assessed as inhibition of CO2 hydration preincubated for 15 mins prior to testing by phenol red ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Egyptian Russian University

Curated by ChEMBL
LigandPNGBDBM50378550(CHEMBL4167551)
Affinity DataKi:  39nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition of CO2 hydration preincubated for 15 mins prior to testing by phenol red ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Egyptian Russian University

Curated by ChEMBL
LigandPNGBDBM50378550(CHEMBL4167551)
Affinity DataKi:  747nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 assessed as inhibition of CO2 hydration preincubated for 15 mins prior to testing by phenol red ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Egyptian Russian University

Curated by ChEMBL
LigandPNGBDBM50378550(CHEMBL4167551)
Affinity DataKi:  2.81E+3nMAssay Description:Inhibition of recombinant human carbonic anhydrase 4 assessed as inhibition of CO2 hydration preincubated for 15 mins prior to testing by phenol red ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed