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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Kelch-like ECH-associated protein 1
(Homo sapiens (Human))
The State University Of New Jersey
Curated by
ChEMBL
Ligand
BDBM50593815
(CHEMBL5184245)
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Affinity Data
IC50: 14nM
Assay Description:
Inhibition of His-tagged Keap1 kelch domain/Nrf2 (unknown origin) protein-protein interaction using FITC-LDEETGEFL-NH2 peptide as substrate preincuba...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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PC cid
PC sid
In Depth
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PubMed
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Target
Kelch-like ECH-associated protein 1
(Homo sapiens (Human))
The State University Of New Jersey
Curated by
ChEMBL
Ligand
BDBM50593815
(CHEMBL5184245)
Copy SMILES
Copy InChI
Affinity Data
IC50: 65nM
Assay Description:
Inhibition of recombinant human Keap1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells/Nrf2 (unknown origin) pr...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI